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KINLYTIC (UROKINASE FOR INJECTION) 250000 UNIT — DIN 00749702

UROKINASE : 250000 UNIT · MICROBIX BIOSYSTEMS INC · POWDER FOR SOLUTION · wholesale supply in Canada

Health Canada status: CANCELLED POST MARKET

What is KINLYTIC (UROKINASE FOR INJECTION)?

KINLYTIC (UROKINASE FOR INJECTION) 250000 UNIT contains UROKINASE : 250000 UNIT. It is listed in the Health Canada Drug Product Database under DIN 00749702, held by MICROBIX BIOSYSTEMS INC, supplied as POWDER FOR SOLUTION for INTRAVENOUS administration. Health Canada currently lists it as cancelled post market, status dated 28-Oct-2009. This Drug Identification Number is no longer authorized for sale in Canada, so Nexara does not supply it. The record is kept here because buyers still meet the number on old formularies, purchase orders and tender documents; Nexara can help identify an authorized alternative.

What is KINLYTIC (UROKINASE FOR INJECTION) used for?

Lysis of acute massive pulmonary emboli; coronary artery thrombosis; peripheral arterial and graft thromboembolic occlusion; restoration of patency to intravenous catheters.

Authorized indication as written in the Health Canada product monograph. For healthcare professionals and licensed purchasers; this is not medical advice.

Is there a generic Urokinase in Canada, and who makes it?

Every market authorization holder with a Canadian DIN for this molecule, and how many of their listings Health Canada currently shows as marketed.

Only one market authorization holder has a Canadian DIN containing Urokinase — 2 DINs, of which 0 are currently marketed. There is no second Canadian source today, so a supply interruption on this holder has no domestic substitute at the same molecule.

Market authorization holderDINsMarketedBrand namesPosition
MICROBIX BIOSYSTEMS INC20KINLYTIC (UROKINASE FOR INJECTION), KINLYTIC OPEN-CATHNo marketed DIN

Health Canada’s Drug Product Database does not flag which listing is the originator and which are subsequent-entry products, so Nexara does not label them here. Interchangeability is determined provincially, not federally — confirm for your province before a formulary switch. Nexara can confirm which of these is actually obtainable, and on what lead time, per order.

How is it supplied and stored?

Pack configuration, storage class and the handling constraints that drive cold-chain planning. One DIN can cover more than one pack size, and the pack — not the DIN — is what gets priced, shipped and invoiced.

Strength on the label250000 UNIT
Dosage formPOWDER FOR SOLUTION
RouteINTRAVENOUS
Pack configuration (monograph)Vials containing 250,000 IU or 1,000,000 IU of urokinase. Also available as KINLYTIC OPEN-CATH in 5,000 IU or 9,000 IU vials.
StorageStore powder at 2° - 30°C. Reconstitute immediately before use; contains no preservatives.

Pack detail is kept as a regulatory record. This DIN is no longer authorized for sale in Canada, so Nexara does not quote this pack.

Substance and classification

Active substanceUrokinase
ATC codeB01AD04
AHFS class20:12.20
Biosimilar biologicNo

Health Canada record and identifiers

The regulatory facts straight from the Drug Product Database, plus every identifier form Nexara accepts on a purchase order. A DIN written without its leading zeros is the commonest reason an order line fails to match.

DIN (8-digit, as used in ordering)00749702
DIN (unpadded, as printed on some documents)749702
Brand nameKINLYTIC (UROKINASE FOR INJECTION)
Generic / active ingredientUROKINASE : 250000 UNIT
Market authorization holderMICROBIX BIOSYSTEMS INC
Health Canada scheduleSchedule D
ATC codeB01AD04
ATC anatomical main groupB — Blood and blood-forming organs
ATC therapeutic subgroupB01AD
Current statusCANCELLED POST MARKET
Status date28-Oct-2009
Original market date1988-12-31 00:00:00
Status sourceLive Health Canada DPD sync

Verify on the primary sources

Health Canada DPD record Approved product monograph (PDF)

How is it administered?

Pulmonary Embolism: 4,400 IU/kg priming dose over 10 min, then 4,400 IU/kg/hr for 12 hours. Also used for coronary artery thrombi, peripheral arterial occlusion, and I.V. catheter clearance.

Included because it drives pack selection and wastage. Consult the monograph.

Contraindications

Active internal bleeding, history of CVA, recent intracranial/intraspinal surgery or trauma, intracranial neoplasm, aneurysm, bleeding diathesis, severe uncontrolled hypertension, aortic dissection.

Warnings and precautions

Potential for transmission of infectious agents (human source material). High risk of bleeding; avoid invasive procedures. Monitor for cholesterol embolization and reperfusion arrhythmias.

What can be used instead?

Alternatives on every axis a buyer actually considers — the same molecule in another presentation, the same class, an adjacent class, or a fixed-dose combination. Every row is led by the marketed DIN count, because that is what can be bought this week.

1 · Same molecule, other Canadian presentations

0 of 2 Canadian DINs for this molecule are currently marketed. Marketed products are listed first.

ProductStrengthFormHolderHealth Canada statusDIN
KINLYTIC OPEN-CATH5000 UNITPOWDER FOR SOLUTIONMICROBIX BIOSYSTEMS INCCANCELLED POST MARKET00886777

2 · Same class — other molecules in ATC B01AD

MoleculeCanadian brandsDINsMarketedSourceable
AlteplaseACTIVASE RT-PA · ACTIVASE RT-PA INJ · CATHFLO · LYSATEC RT - PA53Yes
TenecteplaseTNKASE11Yes
StreptokinaseKABIKINASE - PWS 1500000UNITS/VIAL · KABIKINASE - PWS 250000 UNIT/VIAL · KABIKINASE - PWS 750000UNITS/VIAL · STREPTASE · +3 more90Not in Canada
UrokinaseKINLYTIC (UROKINASE FOR INJECTION) · KINLYTIC OPEN-CATH20Not in Canada
Drotrecogin AlfaXIGRIS (20MG/VIAL) · XIGRIS (5MG/VIAL)20Not in Canada
ReteplaseRETAVASE10Not in Canada
AnistreplaseEMINASE 30 UNITS10Not in Canada
AncrodVIPRINEX10Not in Canada

A molecule with zero marketed DINs cannot be sourced domestically, however many approvals it holds — if one of these sits on a formulary or in an older protocol, that is the line to check.

3 · Adjacent classes in ATC B01A

ATC subgroupMoleculesDINsMarketed
B01AFApixaban · Edoxaban · Rivaroxaban159121
B01ABAntithrombin · Dalteparin · Danaparoid · Enoxaparin · Heparin · +3 more12882
B01ACAbciximab · Acetylsalicylic Acid · Cangrelor · Clopidogrel · Combinations · +10 more15866
B01AAAcenocoumarol · Warfarin6216
B01AEArgatroban · Bivalirudin · Dabigatran Etexilate · Lepirudin1811
B01AXCaplacizumab · Defibrotide · Fondaparinux105

Not clinical advice. These tables describe what can be supplied in Canada, not what should be prescribed. Substitution within or across classes is a prescriber and pharmacist decision, and interchangeability is determined provincially.

Can this still be bought in Canada?

No. This Drug Identification Number is cancelled post market in Health Canada's Drug Product Database, so the product is no longer authorized for sale in Canada and Nexara does not supply it. This page is kept as a regulatory record.

If you are looking for a current equivalent, the alternatives above list every product sharing this therapeutic class, with the marketed ones first. Ask us to source an alternative

Ordering questions

Who can buy this from Nexara?

Licensed entities only. Nexara holds Health Canada establishment licence DEL 3-002896-A and ships only to a licensed address. Patients and unlicensed buyers are routed to a partner pharmacy.

Is there a minimum order?

Yes, set per product line and per pack multiple rather than on the order total, so you are never asked to buy a part-pack. The minimum for this line is confirmed with your quote.

What is the lead time?

Confirmed per order at quotation, and it depends on current stock position and whether the product is in shortage.

Why is there no price on this page?

Nexara quotes a delivered Canadian price per order, against a verified licence. Foreign list prices are published on incompatible bases and are not a guide to what any buyer can obtain here, so this page shows which markets list the molecule and on what basis, and nothing more.

Can Nexara supply this for a clinical trial?

Yes — comparator and background-therapy supply, including sourcing from other markets where a Canadian pack will not satisfy the protocol. Clinical trial supply.

Sources and disclaimer

Product data sourced from the Health Canada Drug Product Database and the approved product monograph (PDF). Health Canada status reconciled against the live DPD sync. Last reviewed 10 Sep 2026.

Nothing on this page is medical advice. Nexara Health is a licensed wholesale distributor and supplies licensed entities only; consumer orders are routed to a partner pharmacy. Alternatives tables describe supply, not clinical equivalence.

Health Canada Drug Product Database (DPD), DIN 00749702. Last reviewed 2026-09-10. Nexara Health is a licensed wholesaler and supplies licensed entities only; consumer orders are routed to a partner pharmacy.